Schrader, Jil

The inhibition mechanism of human 20S proteasomes enables next-generation inhibitor design. [electronic resource] - Science (New York, N.Y.) Aug 2016 - 594-8 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1095-9203

10.1126/science.aaf8993 doi


Antineoplastic Agents--chemistry
Biocatalysis--drug effects
Boron Compounds--chemistry
Boronic Acids--chemistry
Bortezomib--chemistry
Catalytic Domain--drug effects
Crystallography, X-Ray
Drug Design
Glycine--analogs & derivatives
Humans
Proteasome Endopeptidase Complex--chemistry
Proteasome Inhibitors--chemistry
Protein Conformation
Threonine--analogs & derivatives