Schrader, Jil The inhibition mechanism of human 20S proteasomes enables next-generation inhibitor design. [electronic resource] - Science (New York, N.Y.) Aug 2016 - 594-8 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1095-9203 Standard No.: 10.1126/science.aaf8993 doi Subjects--Topical Terms: Antineoplastic Agents--chemistryBiocatalysis--drug effectsBoron Compounds--chemistryBoronic Acids--chemistryBortezomib--chemistryCatalytic Domain--drug effectsCrystallography, X-RayDrug DesignGlycine--analogs & derivativesHumansProteasome Endopeptidase Complex--chemistryProteasome Inhibitors--chemistryProtein ConformationThreonine--analogs & derivatives