TY - GEN AU - Stanton,Richard A AU - Lu,Xiao AU - Detorio,Mervi AU - Montero,Catherine AU - Hammond,Emily T AU - Ehteshami,Maryam AU - Domaoal,Robert A AU - Nettles,James H AU - Feraud,Michel AU - Schinazi,Raymond F TI - Discovery, characterization, and lead optimization of 7-azaindole non-nucleoside HIV-1 reverse transcriptase inhibitors SN - 1464-3405 PY - 2017///0726 KW - Animals KW - Binding Sites KW - Cell Survival KW - drug effects KW - Chlorocebus aethiops KW - Drug Evaluation, Preclinical KW - HIV Reverse Transcriptase KW - antagonists & inhibitors KW - HIV-1 KW - Humans KW - Indoles KW - chemistry KW - Molecular Docking Simulation KW - Mutagenesis, Site-Directed KW - Protein Binding KW - Protein Structure, Tertiary KW - Reverse Transcriptase Inhibitors KW - Vero Cells N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2016.06.065 ER -