Stanton, Richard A
Discovery, characterization, and lead optimization of 7-azaindole non-nucleoside HIV-1 reverse transcriptase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters 08 2016
- 4101-5 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2016.06.065 doi
Animals
Binding Sites
Cell Survival--drug effects
Chlorocebus aethiops
Drug Evaluation, Preclinical
HIV Reverse Transcriptase--antagonists & inhibitors
HIV-1--drug effects
Humans
Indoles--chemistry
Molecular Docking Simulation
Mutagenesis, Site-Directed
Protein Binding
Protein Structure, Tertiary
Reverse Transcriptase Inhibitors--chemistry
Vero Cells