Temple, Kayla J

Exploration of GGTase-I substrate requirements. Part 1: Synthesis and biochemical evaluation of novel aryl-modified geranylgeranyl diphosphate analogs. [electronic resource] - Bioorganic & medicinal chemistry letters 08 2016 - 3499-502 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1464-3405

10.1016/j.bmcl.2016.06.034 doi


Alkyl and Aryl Transferases--antagonists & inhibitors
Animals
Dose-Response Relationship, Drug
Enzyme Inhibitors--chemical synthesis
Humans
Molecular Structure
Polyisoprenyl Phosphates--chemical synthesis
Structure-Activity Relationship