Johansson, Catrine

Structural analysis of human KDM5B guides histone demethylase inhibitor development. [electronic resource] - Nature chemical biology 07 2016 - 539-45 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1552-4469

10.1038/nchembio.2087 doi


Antineoplastic Agents--chemistry
Cell Proliferation--drug effects
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemistry
Histone Demethylases--antagonists & inhibitors
Humans
Jumonji Domain-Containing Histone Demethylases--chemistry
Models, Molecular
Multiple Myeloma--drug therapy
Nuclear Proteins--chemistry
Protein Conformation
Repressor Proteins--chemistry
Structure-Activity Relationship