Johansson, Catrine Structural analysis of human KDM5B guides histone demethylase inhibitor development. [electronic resource] - Nature chemical biology 07 2016 - 539-45 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1552-4469 Standard No.: 10.1038/nchembio.2087 doi Subjects--Topical Terms: Antineoplastic Agents--chemistryCell Proliferation--drug effectsDrug Screening Assays, AntitumorEnzyme Inhibitors--chemistryHistone Demethylases--antagonists & inhibitorsHumansJumonji Domain-Containing Histone Demethylases--chemistryModels, MolecularMultiple Myeloma--drug therapyNuclear Proteins--chemistryProtein ConformationRepressor Proteins--chemistryStructure-Activity Relationship