Targeting IκB Kinase β/NF-κB Signaling in Human Prostate Cancer by a Novel IκB Kinase β Inhibitor CmpdA. [electronic resource]
- Molecular cancer therapeutics 07 2016
- 1504-14 p. digital
Publication Type: Journal Article
1538-8514
10.1158/1535-7163.MCT-15-0999 doi
Animals Antineoplastic Agents--pharmacology Apoptosis--drug effects Cell Line, Tumor Cell Movement--genetics Cell Transformation, Neoplastic--drug effects Disease Models, Animal Docetaxel Drug Synergism Epithelial-Mesenchymal Transition--genetics Gene Knockdown Techniques Humans I-kappa B Kinase--genetics Male Mechanistic Target of Rapamycin Complex 1 Mice Multiprotein Complexes--metabolism NF-kappa B--genetics Neoplastic Stem Cells--drug effects Phosphorylation Prostatic Neoplasms--genetics Protein Kinase Inhibitors--pharmacology Proto-Oncogene Proteins c-akt--metabolism Signal Transduction--drug effects TOR Serine-Threonine Kinases--metabolism Taxoids--pharmacology Xenograft Model Antitumor Assays