Benoist, Guillemette E

Pharmacokinetic Aspects of the Two Novel Oral Drugs Used for Metastatic Castration-Resistant Prostate Cancer: Abiraterone Acetate and Enzalutamide. [electronic resource] - Clinical pharmacokinetics 11 2016 - 1369-1380 p. digital

Publication Type: Journal Article; Review

1179-1926

10.1007/s40262-016-0403-6 doi


Abiraterone Acetate--pharmacokinetics
Antineoplastic Agents--pharmacokinetics
Area Under Curve
Benzamides
Cytochrome P-450 Enzyme System--drug effects
Dose-Response Relationship, Drug
Drug Interactions
Enzyme Induction--drug effects
Fasting
Half-Life
Humans
Liver Failure--metabolism
Male
Metabolic Clearance Rate
Nitriles
Phenylthiohydantoin--analogs & derivatives
Prostatic Neoplasms, Castration-Resistant--drug therapy
Receptors, Androgen--drug effects