Optimizing the macrocyclic diterpenic core toward the reversal of multidrug resistance in cancer. [electronic resource]
- Future medicinal chemistry 04 2016
- 629-45 p. digital
Publication Type: Journal Article
1756-8927
10.4155/fmc.16.11 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Animals Antineoplastic Agents, Phytogenic--chemistry Cell Line, Tumor Diterpenes--chemistry Drug Resistance, Multiple--drug effects Drug Resistance, Neoplasm--drug effects Drug Screening Assays, Antitumor Euphorbia--chemistry Humans Macrocyclic Compounds--chemistry Mice Molecular Conformation Quantitative Structure-Activity Relationship