Ghandi, Mehdi

One-pot synthesis and sigma receptor binding studies of novel spirocyclic-2,6-diketopiperazine derivatives. [electronic resource] - Bioorganic & medicinal chemistry letters 06 2016 - 2676-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2016.04.010 doi


Animals
Binding Sites--drug effects
Diketopiperazines--chemical synthesis
Dose-Response Relationship, Drug
Guinea Pigs
Humans
Molecular Structure
Rats
Receptors, sigma--antagonists & inhibitors
Structure-Activity Relationship
Sigma-1 Receptor