Ghandi, Mehdi
One-pot synthesis and sigma receptor binding studies of novel spirocyclic-2,6-diketopiperazine derivatives. [electronic resource]
- Bioorganic & medicinal chemistry letters 06 2016
- 2676-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2016.04.010 doi
Animals
Binding Sites--drug effects
Diketopiperazines--chemical synthesis
Dose-Response Relationship, Drug
Guinea Pigs
Humans
Molecular Structure
Rats
Receptors, sigma--antagonists & inhibitors
Structure-Activity Relationship
Sigma-1 Receptor