Lamb, David J

BI 1002494, a Novel Potent and Selective Oral Spleen Tyrosine Kinase Inhibitor, Displays Differential Potency in Human Basophils and B Cells. [electronic resource] - The Journal of pharmacology and experimental therapeutics 06 2016 - 554-61 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-0103

10.1124/jpet.116.233155 doi


Administration, Oral
Animals
B-Lymphocytes--drug effects
Basophils--drug effects
Humans
Male
Mast Cells--drug effects
Naphthyridines--administration & dosage
Protein Kinase Inhibitors--administration & dosage
Pyrrolidines--administration & dosage
Pyrrolidinones--administration & dosage
Rats
Syk Kinase--antagonists & inhibitors