McDermott, Lee A
Design and evaluation of novel glutaminase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry Apr 2016
- 1819-39 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
1464-3391
10.1016/j.bmc.2016.03.009 doi
Benzeneacetamides--chemistry
Cell Line, Tumor
Dose-Response Relationship, Drug
Drug Design
Enzyme Inhibitors--chemistry
Glutaminase--antagonists & inhibitors
Humans
Microsomes, Liver--chemistry
Models, Molecular
Molecular Structure
Structure-Activity Relationship
Sulfides--chemistry
Thiadiazoles--chemistry