Cao, Dong

Synthesis, in vitro and in vivo evaluation of novel substituted N-(4-(2-(4-benzylpiperazin-1-yl)ethoxy)phenyl)-N-methyl-quinazolin-4-amines as potent antitumor agents. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2016 - 1931-5 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2016.03.016 doi


Animals
Antineoplastic Agents--chemical synthesis
Apoptosis--drug effects
Cell Cycle Checkpoints--drug effects
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Humans
Liver Neoplasms, Experimental--drug therapy
Mice
Mice, Nude
Molecular Docking Simulation
Molecular Structure
Piperazines--chemical synthesis
Quinazolines--chemical synthesis
Structure-Activity Relationship