Stauffer, Frédéric

Identification of a 5-[3-phenyl-(2-cyclic-ether)-methylether]-4-aminopyrrolo[2,3-d]pyrimidine series of IGF-1R inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2016 - 2065-7 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2016.02.074 doi


Crystallography, X-Ray
Dose-Response Relationship, Drug
Humans
Microsomes, Liver--chemistry
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Pyrimidines--chemical synthesis
Pyrroles--chemical synthesis
Receptor, IGF Type 1--antagonists & inhibitors
Structure-Activity Relationship