Chai, Sergio C

Small-molecule modulators of PXR and CAR. [electronic resource] - Biochimica et biophysica acta 09 2016 - 1141-1154 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Review

0006-3002

10.1016/j.bbagrm.2016.02.013 doi


Animals
Camptothecin--chemistry
Constitutive Androstane Receptor
Coumestrol--chemistry
Energy Metabolism--drug effects
Gene Expression Regulation
Humans
Inactivation, Metabolic--drug effects
Ketoconazole--chemistry
Liver--drug effects
Metformin--chemistry
Pregnane X Receptor
Protein Binding
Receptors, Cytoplasmic and Nuclear--agonists
Receptors, Steroid--agonists
Signal Transduction
Small Molecule Libraries--chemistry
Species Specificity
Substrate Specificity