Development of a Rat Plasma and Brain Extracellular Fluid Pharmacokinetic Model for Bupropion and Hydroxybupropion Based on Microdialysis Sampling, and Application to Predict Human Brain Concentrations. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals May 2016
- 624-33 p. digital
Publication Type: Journal Article
1521-009X
10.1124/dmd.115.068932 doi
Animals Blood-Brain Barrier--metabolism Brain--metabolism Bupropion--analogs & derivatives Dopamine Plasma Membrane Transport Proteins--metabolism Extracellular Fluid--metabolism Humans Male Microdialysis--methods Norepinephrine Plasma Membrane Transport Proteins--metabolism Plasma--metabolism Rats Rats, Sprague-Dawley