Prado, Silvia
Bioavailable inhibitors of HIV-1 RNA biogenesis identified through a Rev-based screen. [electronic resource]
- Biochemical pharmacology May 2016
- 14-28 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
ISSN: 1873-2968
Standard No.: 10.1016/j.bcp.2016.02.007 doi
Subjects--Topical Terms: Anti-HIV Agents--adverse effects Cell Line Cell Survival--drug effects Clomiphene--adverse effects Cyproheptadine--adverse effects Drug Evaluation, Preclinical Gene Expression Regulation, Viral--drug effects Genes, Reporter--drug effects HIV-1--drug effects High-Throughput Screening Assays Humans Peptide Fragments--antagonists & inhibitors Protein Interaction Domains and Motifs RNA Splicing--drug effects RNA, Viral--metabolism Recombinant Proteins--chemistry Response Elements--drug effects Small Molecule Libraries Transcription, Genetic--drug effects rev Gene Products, Human Immunodeficiency Virus--antagonists & inhibitors