Guo, Dong
Molecular Basis of Ligand Dissociation from the Adenosine A2A Receptor. [electronic resource]
- Molecular pharmacology May 2016
- 485-91 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1521-0111
10.1124/mol.115.102657 doi
Adenosine A2 Receptor Antagonists--chemistry
Amino Acid Substitution
Binding Sites
Cell Membrane--chemistry
Databases, Protein
HEK293 Cells
Humans
Hydrogen Bonding
Hydrophobic and Hydrophilic Interactions
Kinetics
Ligands
Models, Molecular
Molecular Conformation
Molecular Dynamics Simulation
Mutation
Radioligand Assay
Receptor, Adenosine A2A--chemistry
Recombinant Proteins--chemistry
Solubility
Triazines--chemistry
Triazoles--chemistry