Design and optimization of tricyclic gamma-secretase modulators. [electronic resource]
- Bioorganic & medicinal chemistry letters Mar 2016
- 1498-502 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2015.06.020 doi
Amyloid Precursor Protein Secretases--antagonists & inhibitors Aniline Compounds--chemical synthesis Animals Dose-Response Relationship, Drug Drug Design Humans Mice Molecular Structure Protease Inhibitors--chemical synthesis Structure-Activity Relationship Triazines--chemical synthesis