TY - GEN AU - Pala,Daniele AU - Rivara,Silvia AU - Mor,Marco AU - Milazzo,Ferdinando Maria AU - Roscilli,Giuseppe AU - Pavoni,Emiliano AU - Giannini,Giuseppe TI - Kinetic analysis and molecular modeling of the inhibition mechanism of roneparstat (SST0001) on human heparanase SN - 1460-2423 PY - 2017///1227 KW - Acidobacteria KW - chemistry KW - Amino Acid Motifs KW - Binding Sites KW - Carbohydrate Sequence KW - Enzyme Inhibitors KW - Fondaparinux KW - Glucuronidase KW - antagonists & inhibitors KW - Heparin KW - analogs & derivatives KW - Humans KW - Kinetics KW - Molecular Docking Simulation KW - Molecular Dynamics Simulation KW - Polysaccharides KW - Protein Binding KW - Protein Conformation, alpha-Helical KW - Protein Conformation, beta-Strand KW - Protein Interaction Domains and Motifs KW - Recombinant Proteins KW - Structural Homology, Protein KW - Substrate Specificity KW - Thermodynamics N1 - Publication Type: Journal Article UR - https://doi.org/10.1093/glycob/cww003 ER -