Pala, Daniele

Kinetic analysis and molecular modeling of the inhibition mechanism of roneparstat (SST0001) on human heparanase. [electronic resource] - Glycobiology 06 2016 - 640-54 p. digital

Publication Type: Journal Article

1460-2423

10.1093/glycob/cww003 doi


Acidobacteria--chemistry
Amino Acid Motifs
Binding Sites
Carbohydrate Sequence
Enzyme Inhibitors--chemistry
Fondaparinux
Glucuronidase--antagonists & inhibitors
Heparin--analogs & derivatives
Humans
Kinetics
Molecular Docking Simulation
Molecular Dynamics Simulation
Polysaccharides--chemistry
Protein Binding
Protein Conformation, alpha-Helical
Protein Conformation, beta-Strand
Protein Interaction Domains and Motifs
Recombinant Proteins--chemistry
Structural Homology, Protein
Substrate Specificity
Thermodynamics