Shu, Shaokun
Response and resistance to BET bromodomain inhibitors in triple-negative breast cancer. [electronic resource]
- Nature Jan 2016
- 413-417 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
1476-4687
10.1038/nature16508 doi
Animals
Azepines--pharmacology
Binding, Competitive--drug effects
Casein Kinase II--metabolism
Cell Cycle Proteins
Cell Line, Tumor
Cell Proliferation--drug effects
Chromatin--genetics
Drug Resistance, Neoplasm--drug effects
Epigenesis, Genetic--drug effects
Female
Gene Expression Regulation, Neoplastic--drug effects
Genome, Human--drug effects
Humans
Mediator Complex Subunit 1--metabolism
Mice
Nuclear Proteins--antagonists & inhibitors
Phosphorylation--drug effects
Phosphoserine--metabolism
Protein Binding--drug effects
Protein Phosphatase 2--metabolism
Protein Structure, Tertiary--drug effects
Proteomics
Transcription Factors--antagonists & inhibitors
Transcription, Genetic--drug effects
Triazoles--pharmacology
Triple Negative Breast Neoplasms--drug therapy
Xenograft Model Antitumor Assays