TY - GEN AU - Goyard,David AU - Kónya,Bálint AU - Chajistamatiou,Aikaterini S AU - Chrysina,Evangelia D AU - Leroy,Jérémy AU - Balzarin,Sophie AU - Tournier,Michel AU - Tousch,Didier AU - Petit,Pierre AU - Duret,Cédric AU - Maurel,Patrick AU - Somsák,László AU - Docsa,Tibor AU - Gergely,Pál AU - Praly,Jean-Pierre AU - Azay-Milhau,Jacqueline AU - Vidal,Sébastien TI - Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition SN - 1768-3254 PY - 2016///1011 KW - Animals KW - Diabetes Mellitus, Experimental KW - drug therapy KW - Diabetes Mellitus, Type 2 KW - Disease Models, Animal KW - Dose-Response Relationship, Drug KW - Enzyme Inhibitors KW - chemical synthesis KW - Glucose KW - analogs & derivatives KW - Glycogen Phosphorylase KW - antagonists & inhibitors KW - Hypoglycemic Agents KW - Isoxazoles KW - Molecular Structure KW - Rats KW - Rats, Zucker KW - Spiro Compounds KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.ejmech.2015.12.004 ER -