Cheng, Jianjun

Further Advances in Optimizing (2-Phenylcyclopropyl)methylamines as Novel Serotonin 2C Agonists: Effects on Hyperlocomotion, Prepulse Inhibition, and Cognition Models. [electronic resource] - Journal of medicinal chemistry Jan 2016 - 578-91 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1520-4804

10.1021/acs.jmedchem.5b01153 doi


Animals
Brain--metabolism
Catalepsy--chemically induced
Central Nervous System Stimulants
Cognition--drug effects
Dextroamphetamine
Drug Design
Drug Evaluation, Preclinical
Ether-A-Go-Go Potassium Channels--antagonists & inhibitors
Female
Humans
Hyperkinesis--chemically induced
Male
Mice
Mice, Inbred C57BL
Microsomes, Liver--metabolism
Prepulse Inhibition--drug effects
Receptor, Serotonin, 5-HT2C--drug effects
Recognition, Psychology--drug effects
Schizophrenia--drug therapy
Schizophrenic Psychology
Serotonin 5-HT2 Receptor Agonists--chemical synthesis
Structure-Activity Relationship
Substrate Specificity