Perez Diaz, Noelia

In silico modelling of prostacyclin and other lipid mediators to nuclear receptors reveal novel thyroid hormone receptor antagonist properties. [electronic resource] - Prostaglandins & other lipid mediators Jan 2016 - 18-27 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1098-8823

10.1016/j.prostaglandins.2015.12.002 doi


Animals
Binding, Competitive--drug effects
Computer Simulation
Dose-Response Relationship, Drug
Epoprostenol--analogs & derivatives
Humans
Ligands
Male
Mesenteric Arteries--drug effects
Models, Molecular
Myography--methods
Protein Domains
Rats, Wistar
Receptors, Cytoplasmic and Nuclear--agonists
Receptors, Thyroid Hormone--antagonists & inhibitors
Thiazoles--chemistry
Thyroid Hormone Receptors alpha--antagonists & inhibitors
Thyroid Hormone Receptors beta--antagonists & inhibitors
Triiodothyronine--metabolism
Vasodilation--drug effects