Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. [electronic resource]
- Chemistry & biology Dec 2015
- 1588-96 p. digital
Publication Type: Journal Article
1879-1301
10.1016/j.chembiol.2015.10.013 doi
CREB-Binding Protein--antagonists & inhibitors Drug Design Fluorescence Resonance Energy Transfer Gene Expression Regulation--drug effects Humans Protein Structure, Tertiary RGS Proteins--genetics Small Molecule Libraries--chemistry Transcriptome