Chekler, Eugene L Piatnitski

Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. [electronic resource] - Chemistry & biology Dec 2015 - 1588-96 p. digital

Publication Type: Journal Article

1879-1301

10.1016/j.chembiol.2015.10.013 doi


CREB-Binding Protein--antagonists & inhibitors
Drug Design
Fluorescence Resonance Energy Transfer
Gene Expression Regulation--drug effects
Humans
Protein Structure, Tertiary
RGS Proteins--genetics
Small Molecule Libraries--chemistry
Transcriptome