Nasiri, Hamid R

Thermodynamic profiling of inhibitors of Nrf2:Keap1 interactions. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2016 - 526-529 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2015.11.082 doi


High-Throughput Screening Assays--methods
Kelch-Like ECH-Associated Protein 1--antagonists & inhibitors
NF-E2-Related Factor 2--antagonists & inhibitors
Oxazines--chemistry
Protein Binding
Protein Structure, Quaternary
Pyrrolidines--chemistry
Sulfonamides--chemistry
Temperature
Thermodynamics