The Influence of the 1-(3-Trifluoromethyl-Benzyl)-1H-Pyrazole-4-yl Moiety on the Adenosine Receptors Affinity Profile of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine Derivatives. [electronic resource]
- PloS one 2015
- e0143504 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1932-6203
10.1371/journal.pone.0143504 doi
Animals CHO Cells Cricetinae Cricetulus Humans Models, Molecular Protein Binding Protein Conformation Purinergic P1 Receptor Antagonists--chemistry Pyrazoles--chemistry Pyrimidines--chemistry Receptors, Purinergic P1--chemistry Structure-Activity Relationship