Buontempo, Francesca

Synergistic cytotoxic effects of bortezomib and CK2 inhibitor CX-4945 in acute lymphoblastic leukemia: turning off the prosurvival ER chaperone BIP/Grp78 and turning on the pro-apoptotic NF-κB. [electronic resource] - Oncotarget Jan 2016 - 1323-40 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1949-2553

10.18632/oncotarget.6361 doi


Antineoplastic Agents--pharmacology
Apoptosis--drug effects
Blotting, Western
Bortezomib--pharmacology
Casein Kinase II--antagonists & inhibitors
Cell Line, Tumor
Cell Survival--drug effects
Drug Synergism
Endoplasmic Reticulum Chaperone BiP
Endoplasmic Reticulum Stress--drug effects
Heat-Shock Proteins--metabolism
Humans
Jurkat Cells
Microscopy, Fluorescence
Naphthyridines--pharmacology
Neoplastic Stem Cells--drug effects
Phenazines
Precursor B-Cell Lymphoblastic Leukemia-Lymphoma--blood
Precursor Cell Lymphoblastic Leukemia-Lymphoma--blood
Precursor T-Cell Lymphoblastic Leukemia-Lymphoma--blood
Transcription Factor RelA--metabolism
Unfolded Protein Response--drug effects