Small Molecule T315 Promotes Casitas B-Lineage Lymphoma-Dependent Degradation of Epidermal Growth Factor Receptor via Y1045 Autophosphorylation. [electronic resource]
- American journal of respiratory and critical care medicine Apr 2016
- 753-66 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1535-4970
10.1164/rccm.201502-0250OC doi
Adaptor Proteins, Signal Transducing--drug effects Adenocarcinoma--drug therapy Adenocarcinoma of Lung Afatinib Animals Antineoplastic Agents--adverse effects Blotting, Western Cell Proliferation--drug effects Drug Combinations Drug Resistance, Neoplasm--drug effects Enzyme Assays ErbB Receptors--antagonists & inhibitors Humans Lung Neoplasms--drug therapy Mass Spectrometry Mice Mutation--genetics Protein Kinase Inhibitors--adverse effects Proto-Oncogene Proteins c-cbl--drug effects Quinazolines--adverse effects Real-Time Polymerase Chain Reaction Tumor Cells, Cultured Xenograft Model Antitumor Assays