Manda, Sudhakar

Discovery of a marine-derived bis-indole alkaloid fascaplysin, as a new class of potent P-glycoprotein inducer and establishment of its structure-activity relationship. [electronic resource] - European journal of medicinal chemistry Jan 2016 - 1-11 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1768-3254

10.1016/j.ejmech.2015.10.049 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Biological Products--chemistry
Cell Line
Chemistry Techniques, Synthetic
Cholinesterase Inhibitors--chemistry
Drug Evaluation, Preclinical--methods
Humans
Indoles--chemical synthesis
Molecular Docking Simulation
Solubility
Structure-Activity Relationship