Discovery of a marine-derived bis-indole alkaloid fascaplysin, as a new class of potent P-glycoprotein inducer and establishment of its structure-activity relationship. [electronic resource]
- European journal of medicinal chemistry Jan 2016
- 1-11 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2015.10.049 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism Biological Products--chemistry Cell Line Chemistry Techniques, Synthetic Cholinesterase Inhibitors--chemistry Drug Evaluation, Preclinical--methods Humans Indoles--chemical synthesis Molecular Docking Simulation Solubility Structure-Activity Relationship