TY  - GEN
AU  - Johansson,Henrik
AU  - Boesgaard,Michael Worch
AU  - Nørskov-Lauritsen,Lenea
AU  - Larsen,Inna
AU  - Kuhne,Sebastiaan
AU  - Gloriam,David E
AU  - Bräuner-Osborne,Hans
AU  - Sejer Pedersen,Daniel
TI  - Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2-Phenylindole Privileged Structure Scaffold
SN  - 1520-4804
PY  - 2016///0314
KW  - Animals
KW  - CHO Cells
KW  - Cell Line
KW  - Cricetinae
KW  - Cricetulus
KW  - Cyclization
KW  - Drug Design
KW  - Goldfish
KW  - HEK293 Cells
KW  - Humans
KW  - Indoles
KW  - chemical synthesis
KW  - Inosine Monophosphate
KW  - metabolism
KW  - Ligands
KW  - Mice
KW  - Rats
KW  - Receptors, G-Protein-Coupled
KW  - antagonists & inhibitors
KW  - Structure-Activity Relationship
KW  - Transfection
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1021/acs.jmedchem.5b01254
ER  -