Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2-Phenylindole Privileged Structure Scaffold. [electronic resource]
- Journal of medicinal chemistry Nov 2015
- 8938-51 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/acs.jmedchem.5b01254 doi
Animals CHO Cells Cell Line Cricetinae Cricetulus Cyclization Drug Design Goldfish HEK293 Cells Humans Indoles--chemical synthesis Inosine Monophosphate--metabolism Ligands Mice Rats Receptors, G-Protein-Coupled--antagonists & inhibitors Structure-Activity Relationship Transfection