Johansson, Henrik

Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2-Phenylindole Privileged Structure Scaffold. [electronic resource] - Journal of medicinal chemistry Nov 2015 - 8938-51 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.5b01254 doi


Animals
CHO Cells
Cell Line
Cricetinae
Cricetulus
Cyclization
Drug Design
Goldfish
HEK293 Cells
Humans
Indoles--chemical synthesis
Inosine Monophosphate--metabolism
Ligands
Mice
Rats
Receptors, G-Protein-Coupled--antagonists & inhibitors
Structure-Activity Relationship
Transfection