3-Halo Chloroquine Derivatives Overcome Plasmodium falciparum Chloroquine Resistance Transporter-Mediated Drug Resistance in P. falciparum. [electronic resource]
- Antimicrobial agents and chemotherapy Dec 2015
- 7891-3 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1098-6596
10.1128/AAC.01139-15 doi
Antimalarials--chemical synthesis Chloroquine--analogs & derivatives Dose-Response Relationship, Drug Drug Resistance--drug effects Gene Expression Halogenation Membrane Transport Proteins--genetics Parasitic Sensitivity Tests Plasmodium falciparum--drug effects Polymorphism, Genetic Protozoan Proteins--antagonists & inhibitors