TY  - GEN
AU  - Goswami,Rajeev
AU  - Wohlfahrt,Gerd
AU  - Törmäkangas,Olli
AU  - Moilanen,Anu
AU  - Lakshminarasimhan,Anirudha
AU  - Nagaraj,Jwala
AU  - Arumugam,Karthikeyan N
AU  - Mukherjee,Subhendu
AU  - Chacko,Anita R
AU  - Krishnamurthy,Narasimha R
AU  - Jaleel,Mahaboobi
AU  - Palakurthy,Rajendra K
AU  - Samiulla,Dodheri S
AU  - Ramachandra,Murali
TI  - Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors
SN  - 1464-3405
PY  - 2016///0628
KW  - Animals
KW  - Antineoplastic Agents
KW  - chemical synthesis
KW  - Cell Line, Tumor
KW  - Cell Movement
KW  - drug effects
KW  - Cyclohexanes
KW  - Humans
KW  - Indoles
KW  - Mice
KW  - Microsomes, Liver
KW  - metabolism
KW  - Molecular Docking Simulation
KW  - Neoplasm Invasiveness
KW  - Pyridines
KW  - Serine Endopeptidases
KW  - Serine Proteinase Inhibitors
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1016/j.bmcl.2015.09.042
ER  -