Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors. [electronic resource]
- ACS chemical biology Dec 2015
- 2716-24 p. digital
Publication Type: Journal Article
1554-8937
10.1021/acschembio.5b00334 doi
Computer Simulation Cytosol--chemistry Drug Delivery Systems Drug Evaluation, Preclinical Enzyme Inhibitors--chemical synthesis Extracellular Space--enzymology Inhibitory Concentration 50 Insulin Antagonists--pharmacology Insulysin--antagonists & inhibitors Models, Biological Molecular Structure Structure-Activity Relationship Sulfhydryl Compounds--chemistry