Abdul-Hay, Samer O

Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors. [electronic resource] - ACS chemical biology Dec 2015 - 2716-24 p. digital

Publication Type: Journal Article

1554-8937

10.1021/acschembio.5b00334 doi


Computer Simulation
Cytosol--chemistry
Drug Delivery Systems
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Extracellular Space--enzymology
Inhibitory Concentration 50
Insulin Antagonists--pharmacology
Insulysin--antagonists & inhibitors
Models, Biological
Molecular Structure
Structure-Activity Relationship
Sulfhydryl Compounds--chemistry