Reese, Melinda J
Drug interaction profile of the HIV integrase inhibitor cabotegravir: assessment from in vitro studies and a clinical investigation with midazolam. [electronic resource]
- Xenobiotica; the fate of foreign compounds in biological systems 2016
- 445-56 p. digital
Publication Type: Clinical Trial, Phase I; Journal Article; Research Support, Non-U.S. Gov't
ISSN: 1366-5928
Standard No.: 10.3109/00498254.2015.1081993 doi
Subjects--Topical Terms: ATP-Binding Cassette Transporters--metabolism Administration, Oral Adolescent Adult Aged Animals Anti-HIV Agents--administration & dosage Area Under Curve Cytochrome P-450 CYP3A--chemistry Dogs Dose-Response Relationship, Drug Drug Interactions Female HIV Infections--drug therapy HIV Integrase Inhibitors--chemistry Hepatocytes--drug effects Humans Inhibitory Concentration 50 Madin Darby Canine Kidney Cells Male Midazolam--administration & dosage Middle Aged Organic Anion Transport Protein 1--antagonists & inhibitors Organic Anion Transporters--metabolism Organic Anion Transporters, Sodium-Independent--antagonists & inhibitors Pyridones--administration & dosage Young Adult