Reese, Melinda J

Drug interaction profile of the HIV integrase inhibitor cabotegravir: assessment from in vitro studies and a clinical investigation with midazolam. [electronic resource] - Xenobiotica; the fate of foreign compounds in biological systems 2016 - 445-56 p. digital

Publication Type: Clinical Trial, Phase I; Journal Article; Research Support, Non-U.S. Gov't

1366-5928

10.3109/00498254.2015.1081993 doi


ATP-Binding Cassette Transporters--metabolism
Administration, Oral
Adolescent
Adult
Aged
Animals
Anti-HIV Agents--administration & dosage
Area Under Curve
Cytochrome P-450 CYP3A--chemistry
Dogs
Dose-Response Relationship, Drug
Drug Interactions
Female
HIV Infections--drug therapy
HIV Integrase Inhibitors--chemistry
Hepatocytes--drug effects
Humans
Inhibitory Concentration 50
Madin Darby Canine Kidney Cells
Male
Midazolam--administration & dosage
Middle Aged
Organic Anion Transport Protein 1--antagonists & inhibitors
Organic Anion Transporters--metabolism
Organic Anion Transporters, Sodium-Independent--antagonists & inhibitors
Pyridones--administration & dosage
Young Adult