Selection of High-Affinity Peptidic Serine Protease Inhibitors with Increased Binding Entropy from a Back-Flip Library of Peptide-Protease Fusions. [electronic resource]
- Journal of molecular biology Sep 2015
- 3110-22 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1089-8638
10.1016/j.jmb.2015.08.005 doi
Amino Acid Sequence Animals Cell Line Crystallography, X-Ray Drug Discovery Entropy Humans Mice Molecular Sequence Data Peptide Library Peptides, Cyclic--chemistry Protein Conformation Recombinant Fusion Proteins--chemistry Serine Endopeptidases--chemistry Serine Proteinase Inhibitors--chemistry Urokinase-Type Plasminogen Activator--antagonists & inhibitors