Sørensen, Hans Peter

Selection of High-Affinity Peptidic Serine Protease Inhibitors with Increased Binding Entropy from a Back-Flip Library of Peptide-Protease Fusions. [electronic resource] - Journal of molecular biology Sep 2015 - 3110-22 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1089-8638

10.1016/j.jmb.2015.08.005 doi


Amino Acid Sequence
Animals
Cell Line
Crystallography, X-Ray
Drug Discovery
Entropy
Humans
Mice
Molecular Sequence Data
Peptide Library
Peptides, Cyclic--chemistry
Protein Conformation
Recombinant Fusion Proteins--chemistry
Serine Endopeptidases--chemistry
Serine Proteinase Inhibitors--chemistry
Urokinase-Type Plasminogen Activator--antagonists & inhibitors