Synthesis, Biological, and Computational Evaluation of Novel 1,3,5-Substituted Indolin-2-one Derivatives as Inhibitors of Src Tyrosine Kinase. [electronic resource]
- Archiv der Pharmazie Oct 2015
- 715-29 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
1521-4184
10.1002/ardp.201500109 doi
Drug Design Hydrogen Bonding Imatinib Mesylate--pharmacology Indoles--chemical synthesis Molecular Docking Simulation Molecular Targeted Therapy Phosphorylation Phosphotyrosine--metabolism Protein Conformation Protein Kinase Inhibitors--chemical synthesis Structure-Activity Relationship src-Family Kinases--antagonists & inhibitors