TY - GEN AU - Savi,Lida AU - Brindisi,Margherita AU - Alfano,Gloria AU - Butini,Stefania AU - La Pietra,Valeria AU - Novellino,Ettore AU - Marinelli,Luciana AU - Lossani,Andrea AU - Focher,Federico AU - Cavella,Caterina AU - Campiani,Giuseppe AU - Gemma,Sandra TI - Site-directed Mutagenesis of Key Residues Unveiled a Novel Allosteric Site on Human Adenosine Kinase for Pyrrolobenzoxa(thia)zepinone Non-Nucleoside Inhibitors SN - 1747-0285 PY - 2016///1213 KW - Adenosine Kinase KW - metabolism KW - Allosteric Site KW - Azepines KW - pharmacology KW - Humans KW - Mutagenesis, Site-Directed KW - Nucleosides KW - antagonists & inhibitors N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1111/cbdd.12630 ER -