TY - GEN AU - Feng,Yu AU - Degen,David AU - Wang,Xinyue AU - Gigliotti,Matthew AU - Liu,Shuang AU - Zhang,Yu AU - Das,Deepankar AU - Michalchuk,Trevor AU - Ebright,Yon W AU - Talaue,Meliza AU - Connell,Nancy AU - Ebright,Richard H TI - Structural Basis of Transcription Inhibition by CBR Hydroxamidines and CBR Pyrazoles SN - 1878-4186 PY - 2016///0520 KW - Amidines KW - chemistry KW - Amino Acid Sequence KW - Animals KW - Anti-Bacterial Agents KW - Binding Sites KW - Chlorocebus aethiops KW - Crystallography, X-Ray KW - DNA-Directed RNA Polymerases KW - antagonists & inhibitors KW - Drug Synergism KW - Escherichia coli KW - drug effects KW - Escherichia coli Proteins KW - HeLa Cells KW - Humans KW - Hydroxylamines KW - Ligands KW - Models, Molecular KW - Molecular Sequence Data KW - Mycobacterium tuberculosis KW - Protein Binding KW - Protein Structure, Secondary KW - Protein Structure, Tertiary KW - Pyrazoles KW - Recombinant Proteins KW - Sequence Alignment KW - Transcription, Genetic KW - Vero Cells N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural UR - https://doi.org/10.1016/j.str.2015.06.009 ER -