Structural Basis of Transcription Inhibition by CBR Hydroxamidines and CBR Pyrazoles. [electronic resource]
- Structure (London, England : 1993) Aug 2015
- 1470-1481 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1878-4186
10.1016/j.str.2015.06.009 doi
Amidines--chemistry Amino Acid Sequence Animals Anti-Bacterial Agents--chemistry Binding Sites Chlorocebus aethiops Crystallography, X-Ray DNA-Directed RNA Polymerases--antagonists & inhibitors Drug Synergism Escherichia coli--drug effects Escherichia coli Proteins--antagonists & inhibitors HeLa Cells Humans Hydroxylamines--chemistry Ligands Models, Molecular Molecular Sequence Data Mycobacterium tuberculosis--drug effects Protein Binding Protein Structure, Secondary Protein Structure, Tertiary Pyrazoles--chemistry Recombinant Proteins--chemistry Sequence Alignment Transcription, Genetic--drug effects Vero Cells