Uncovering Molecular Bases Underlying Bone Morphogenetic Protein Receptor Inhibitor Selectivity. [electronic resource]
- PloS one 2015
- e0132221 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
1932-6203
10.1371/journal.pone.0132221 doi
Activin Receptors, Type I--antagonists & inhibitors Adenosine Triphosphate--metabolism Amino Acid Motifs Amino Acid Substitution Binding Sites--drug effects Bone Morphogenetic Protein Receptors, Type I--antagonists & inhibitors Crystallography, X-Ray Drug Design Humans Ligands Molecular Docking Simulation Molecular Dynamics Simulation Molecular Structure Point Mutation Protein Conformation Protein Kinase Inhibitors--chemistry Protein Serine-Threonine Kinases--antagonists & inhibitors Protein Structure, Tertiary Pyrazoles--chemistry Pyrimidines--chemistry Quinolines--chemistry Receptor, Transforming Growth Factor-beta Type I Receptors, Transforming Growth Factor beta--antagonists & inhibitors Substrate Specificity Vascular Endothelial Growth Factor Receptor-2--antagonists & inhibitors