A New VMAT-2 Inhibitor NBI-641449 in the Treatment of Huntington Disease. [electronic resource]
- CNS neuroscience & therapeutics Aug 2015
- 662-71 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1755-5949
10.1111/cns.12425 doi
3,4-Dihydroxyphenylacetic Acid--metabolism Animals Cell Survival--drug effects Corpus Striatum--drug effects DNA-Binding Proteins Disease Models, Animal Dopamine--metabolism Dopamine and cAMP-Regulated Phosphoprotein 32--metabolism Dose-Response Relationship, Drug Female Homovanillic Acid--metabolism Huntington Disease--drug therapy Mice, Transgenic Motor Activity--drug effects Nerve Tissue Proteins--metabolism Neurons--drug effects Neuroprotective Agents--pharmacology Nuclear Proteins--metabolism Serotonin Plasma Membrane Transport Proteins--metabolism Tyrosine 3-Monooxygenase--metabolism Vesicular Monoamine Transport Proteins--antagonists & inhibitors