Tantry, Subramanyam J

Whole cell screen based identification of spiropiperidines with potent antitubercular properties. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2015 - 3234-45 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2015.05.087 doi


Animals
Antitubercular Agents--chemical synthesis
Bacteria--drug effects
Drug Resistance, Bacterial--genetics
Genome, Bacterial
High-Throughput Screening Assays
Hypoxia
Lipids--chemistry
Matrix Metalloproteinase 13--biosynthesis
Mice
Microbial Sensitivity Tests
Mycobacterium tuberculosis--drug effects
Piperidines--chemical synthesis
Spiro Compounds--chemical synthesis
Structure-Activity Relationship