Pugsley, Michael K

An examination of the cardiac actions of PD117,302, a κ-opioid receptor agonist. [electronic resource] - European journal of pharmacology Aug 2015 - 330-40 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1879-0712

10.1016/j.ejphar.2015.06.018 doi


Action Potentials
Animals
Anti-Arrhythmia Agents--metabolism
Arrhythmias, Cardiac--etiology
Binding, Competitive
Cardiac Pacing, Artificial
Cerebellum--drug effects
Coronary Occlusion--complications
Disease Models, Animal
Dose-Response Relationship, Drug
Electrocardiography
Guinea Pigs
Heart Conduction System--drug effects
Heart Rate--drug effects
Heart Ventricles--drug effects
Isolated Heart Preparation
Ligands
Male
Mice, Inbred BALB C
Myocardial Contraction--drug effects
Pain--metabolism
Pain Threshold--drug effects
Potassium Channel Blockers--pharmacology
Potassium Channels--drug effects
Protein Binding
Pyrroles--metabolism
Radioligand Assay
Rats, Sprague-Dawley
Receptors, Opioid, kappa--drug effects
Sodium Channel Blockers--pharmacology
Sodium Channels--drug effects
Thiophenes--metabolism
Ventricular Function, Left--drug effects
Ventricular Pressure--drug effects