TY  - GEN
AU  - Ran,Xu
AU  - Zhao,Yujun
AU  - Liu,Liu
AU  - Bai,Longchuan
AU  - Yang,Chao-Yie
AU  - Zhou,Bing
AU  - Meagher,Jennifer L
AU  - Chinnaswamy,Krishnapriya
AU  - Stuckey,Jeanne A
AU  - Wang,Shaomeng
TI  - Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors
SN  - 1520-4804
PY  - 2015///0914
KW  - Antineoplastic Agents
KW  - chemistry
KW  - Carbolines
KW  - Cell Cycle Proteins
KW  - Cell Line, Tumor
KW  - Crystallography, X-Ray
KW  - Humans
KW  - Leukemia
KW  - drug therapy
KW  - Molecular Docking Simulation
KW  - Nuclear Proteins
KW  - antagonists & inhibitors
KW  - Protein Serine-Threonine Kinases
KW  - RNA-Binding Proteins
KW  - Transcription Factors
N1  - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1021/acs.jmedchem.5b00613
ER  -