Diaminothiazoles evade multidrug resistance in cancer cells and xenograft tumour models and develop transient specific resistance: understanding the basis of broad-spectrum versus specific resistance. [electronic resource]
- Carcinogenesis Aug 2015
- 883-93 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1460-2180
10.1093/carcin/bgv072 doi
ATP Binding Cassette Transporter, Subfamily B--metabolism ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry Animals Antineoplastic Agents--chemistry Cell Line, Tumor--drug effects Drug Resistance, Multiple--drug effects Drug Resistance, Neoplasm--drug effects Female Humans Male Mice, SCID Molecular Docking Simulation Paclitaxel--pharmacology Thiazoles--chemistry Tubulin--chemistry Xenograft Model Antitumor Assays