Winneroski, Leonard L

Preparation and biological evaluation of conformationally constrained BACE1 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry Jul 2015 - 3260-8 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.

1464-3391

10.1016/j.bmc.2015.04.062 doi


Amyloid Precursor Protein Secretases--antagonists & inhibitors
Animals
Aspartic Acid Endopeptidases--antagonists & inhibitors
Brain Chemistry
Bridged Bicyclo Compounds--chemical synthesis
Crystallography, X-Ray
Drug Design
Humans
Mice
Molecular Conformation
Molecular Docking Simulation
Protease Inhibitors--chemical synthesis
Stereoisomerism
Thiazines--chemical synthesis