Winneroski, Leonard L
Preparation and biological evaluation of conformationally constrained BACE1 inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry Jul 2015
- 3260-8 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
1464-3391
10.1016/j.bmc.2015.04.062 doi
Amyloid Precursor Protein Secretases--antagonists & inhibitors
Animals
Aspartic Acid Endopeptidases--antagonists & inhibitors
Brain Chemistry
Bridged Bicyclo Compounds--chemical synthesis
Crystallography, X-Ray
Drug Design
Humans
Mice
Molecular Conformation
Molecular Docking Simulation
Protease Inhibitors--chemical synthesis
Stereoisomerism
Thiazines--chemical synthesis