TY  - GEN
AU  - Makarov,Vadim
AU  - Neres,João
AU  - Hartkoorn,Ruben C
AU  - Ryabova,Olga B
AU  - Kazakova,Elena
AU  - Šarkan,Michal
AU  - Huszár,Stanislav
AU  - Piton,Jérémie
AU  - Kolly,Gaëlle S
AU  - Vocat,Anthony
AU  - Conroy,Trent M
AU  - Mikušová,Katarína
AU  - Cole,Stewart T
TI  - The 8-Pyrrole-Benzothiazinones Are Noncovalent Inhibitors of DprE1 from Mycobacterium tuberculosis
SN  - 1098-6596
PY  - 2016///0412
KW  - Alcohol Oxidoreductases
KW  - antagonists & inhibitors
KW  - Animals
KW  - Antitubercular Agents
KW  - pharmacology
KW  - Bacterial Proteins
KW  - Catalytic Domain
KW  - drug effects
KW  - Disease Models, Animal
KW  - Hep G2 Cells
KW  - Humans
KW  - Male
KW  - Mice
KW  - Mice, Inbred BALB C
KW  - Microbial Sensitivity Tests
KW  - methods
KW  - Mycobacterium tuberculosis
KW  - Piperazines
KW  - Pyridines
KW  - Pyrroles
KW  - Spiro Compounds
KW  - Structure-Activity Relationship
KW  - Thiazines
KW  - Tuberculosis
KW  - drug therapy
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1128/AAC.00778-15
ER  -