D'yakonov, Vladimir A

11-Phenylundeca-5Z,9Z-dienoic Acid: Stereoselective Synthesis and Dual Topoisomerase I/IIα Inhibition. [electronic resource] - Current cancer drug targets 2015 - 504-10 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1873-5576

10.2174/1568009615666150506093155 doi


Antigens, Neoplasm--chemistry
Binding Sites
Catalytic Domain
DNA Topoisomerases, Type I--chemistry
DNA Topoisomerases, Type II--chemistry
DNA-Binding Proteins--antagonists & inhibitors
Drug Design
Fatty Acids, Unsaturated--chemical synthesis
Humans
Molecular Docking Simulation
Protein Binding
Protein Conformation
Structure-Activity Relationship
Topoisomerase I Inhibitors--chemical synthesis
Topoisomerase II Inhibitors--chemical synthesis